產(chǎn)品編號(hào) | D60218 |
英文名稱 | TAK-385 |
中文名稱 | 瑞盧戈利 |
別 名 | RVT-601 |
CAS | 737789-87-6 |
檢測(cè)分子量 | 623.63 |
保存條件 | 2-8℃ |
產(chǎn)品介紹 |
Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. Relugolix possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al |